精细化工中间体2024,Vol.54Issue(4) :10-12,16.DOI:10.19342/j.cnki.issn.1009-9212.2024.04.003

双酰胺类化合物引入环丙基制备新型杀虫剂的研究

Study on Novel Pesticides by Introducing Cyclopropyl Group into Diamide Compounds

高鹏 唐余 陈诗桦 潘彤
精细化工中间体2024,Vol.54Issue(4) :10-12,16.DOI:10.19342/j.cnki.issn.1009-9212.2024.04.003

双酰胺类化合物引入环丙基制备新型杀虫剂的研究

Study on Novel Pesticides by Introducing Cyclopropyl Group into Diamide Compounds

高鹏 1唐余 1陈诗桦 1潘彤1
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作者信息

  • 1. 长沙理工大学化学化工学院,湖南长沙 410000
  • 折叠

摘要

在双酰胺类化合物中引入环丙基的结构改造,旨在通过结构改造,提升双酰胺类杀虫剂的杀虫广谱.以2-氟-3-胺基苯甲酸甲酯为原料制备新型双酰胺类化合物N-[2-溴-4-(1,1,1,2,3,3,3-七氟丙-2-基)-6-三氟甲氧基苯基]-3-[N-(环丙甲基)苯甲酰胺基]-2-氟苯甲酰胺(BCPF).有利于该化合物进一步杀虫药效、作用机制及高效杀虫剂的研究.

Abstract

Structural modification of bisamide compounds by introducing cyclopropyl group to improve the insecticidal broad spectrum and mechanism was studied.A novel biamide compound N-[2-bromo-4-(1,1,1,2,3,3,3-heptafluoropropyl-2-yl)-6-trifluoromethoxy-phenyl]-3-[N-(cyclopropyl methyl)benzoyl]-2-fluorobenzamide(BCPF)was prepared from 2-fluoro-3-amino methyl benzoate as raw material.It is beneficial to further study on the efficacy and mechanism of the compound and the development of efficient pesticides.

关键词

环丙基双酰胺类化合物/2-氟-3-胺基苯甲酸甲酯/2-氟-3-[N-(环丙甲基)苯甲酰胺]苯甲酸/N-[2-溴-4-(1,1,1,2,3,3,3-七氟丙-2-基)-6-三氟甲氧基苯基]-3-[N-(环丙甲基)苯甲酰胺基]-2-氟苯甲酰胺

Key words

bisamide compounds/cyclopropyl groups/novel pesticides/2-fluoro-3-[N-(cyclopropyl methyl)benzamide]benzoic acid/N-[2-bromo-4-(1,1,1,2,3,3,3-heptafluoropropyl-2-yl)-6-trifluoromethoxy-phenyl]-3-[N-(cyclopropyl methyl)benzoyl]-2-fluorobenzamide

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出版年

2024
精细化工中间体
湖南化工研究院

精细化工中间体

CSTPCD
影响因子:0.236
ISSN:1009-9212
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