A method of organocatalytic synthesis of 2-pyridone derivatives has been reported.Using N-substituted 3-hydroxy-2-pyridones and Morita-Baylis-Hillman(MBH)carbonates as raw materials,a series of multifunctional molecules featuring a 2-pyridone moiety were rapidly constructed in 51%-91%yields through nucleophilic amine-catalyzed regioselective O-allylic substitution reaction.Functionalization of OH group on N-substituted 3-hydroxy-2-pyridone compounds could be smoothly realized under the current reaction conditions.
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