首页|Rhodium-Catalyzed N-Arylation Addition of Arylboronic Acids to Ketimines
Rhodium-Catalyzed N-Arylation Addition of Arylboronic Acids to Ketimines
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维普
Herein,we report rhodium catalyzed N-arylation via addition of arylboronic acids to electron-deficient α-iminoesters which can be prepared in high efficiency by using easily accessible β-carbonyl esters.The reaction is highly regiospecific to achieve the N-aryl addi-tion efficiently with up to 99％yield under mild conditions.The corresponding product can be further efficiently converted into indoles and a series of other important building blocks.
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