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Mechanisms of drug solubilization by polar lipids in biorelevant media

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Despite the widespread use of lipid excipients in both academic research and oral formulation development, rational selection guidelines are still missing. In the current study, we aimed to establish a link between the molecular structure of commonly used polar lipids and drug solubilization in biorelevant media.

Oral drug deliveryLipid-based formulation excipientsDrug solubilizationPoorly water-soluble drugs

Katev, Vladimir、Vinarov, Zahari、Tcholakova, Slavka

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Sofia Univ, Fac Chem & Pharm, Dept Chem & Pharmaceut Engn, Sofia 1164, Bulgaria

2021

European journal of pharmaceutical sciences

European journal of pharmaceutical sciences

ISTP
ISSN:0928-0987
年,卷(期):2021.159
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